Projects per year
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Dive into the research topics where Hiroshi Hiasa is active. These topic labels come from the works of this person. Together they form a unique fingerprint.
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Projects and Grants
- 2 Finished
Research output
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Design, synthesis and structure-activity relationships of novel 15-membered macrolides: Quinolone/quinoline-containing sidechains tethered to the C-6 position of azithromycin acylides
Fan, B. Z., Hiasa, H., Lv, W., Brody, S., Yang, Z. Y., Aldrich, C., Cushman, M. & Liang, J. H., May 1 2020, In: European Journal of Medicinal Chemistry. 193, 112222.Research output: Contribution to journal › Article › peer-review
3 Scopus citations -
Identification of an ethyl 5,6-dihydropyrazolo[1,5-c]quinazoline-1-carboxylate as a catalytic inhibitor of DNA gyrase
Aguirre, A. L., Chheda, P. R., Lentz, S. R. C., Held, H. A., Groves, N. P., Hiasa, H. & Kerns, R. J., May 15 2020, In: Bioorganic and Medicinal Chemistry. 28, 10, 115439.Research output: Contribution to journal › Article › peer-review
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Analysis of mutational patterns in quinolone resistance-determining regions of GyrA and ParC of clinical isolates
Ostrer, L., Khodursky, R. F., Johnson, J. R., Hiasa, H. & Khodursky, A. B., Mar 2019, In: International Journal of Antimicrobial Agents. 53, 3, p. 318-324 7 p.Research output: Contribution to journal › Article › peer-review
5 Scopus citations -
Novel N-1 substituted fluoroquinolones inhibit human topoisomerase I activity and exhibit anti-proliferative activity
Oppegard, L. M., Delgado, J. L., Kulkarni, C. A., Towle, T. R., Hart, D. E., Williams, B. P., Lentz, S. R. C., Norris, B., Flory, C. M., Schumacher, R. J., Murry, D. J., Kerns, R. J. & Hiasa, H., Apr 15 2019, In: Investigational New Drugs. 37, 2, p. 378-383 6 p.Research output: Contribution to journal › Article › peer-review
Open Access1 Scopus citations -
Probing structural requirements for human topoisomerase I inhibition by a novel N1-Biphenyl fluoroquinolone
Delgado, J. L., Lentz, S. R. C., Kulkarni, C. A., Chheda, P. R., Held, H. A., Hiasa, H. & Kerns, R. J., Jun 15 2019, In: European Journal of Medicinal Chemistry. 172, p. 109-130 22 p.Research output: Contribution to journal › Article › peer-review
2 Scopus citations